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LSD1-IN-11p
CAS No. 2101951-67-9
LSD1-IN-11p( —— )
Catalog No. M13339 CAS No. 2101951-67-9
LSD1-IN-11p is a reversible LSD1 inhibitor with IC50/Kd of 79/21 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
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Biological Information
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Product NameLSD1-IN-11p
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NoteResearch use only, not for human use.
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Brief DescriptionLSD1-IN-11p is a reversible LSD1 inhibitor with IC50/Kd of 79/21 nM.
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DescriptionLSD1-IN-11p is a reversible LSD1 inhibitor with IC50/Kd of 79/21 nM; upregulates the expression of the surrogate cellular biomarker CD86 (IC50=0.52 uM); has moderate oral bioavailability in mice (F%=38%).
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayChromatin/Epigenetic
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TargetHistone Demethylase
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RecptorHistone Demethylase
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Research Area——
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Indication——
Chemical Information
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CAS Number2101951-67-9
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Formula Weight420.473
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Molecular FormulaC22H24N6O3
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Purity>98% (HPLC)
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Solubility——
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SMILES——
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Chemical Name(R)-4-(3-(3-aminopiperidine-1-carbonyl)-5-((3-ethylisoxazol-5-yl)methoxy)-1H-pyrazol-1-yl)benzonitrile
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Mould DP, et al. Bioorg Med Chem Lett. 2017 Jul 15;27(14):3190-3195.
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