MZ-242

CAS No. 1862238-01-4

MZ-242( MZ242 | MZ242 )

Catalog No. M12877 CAS No. 1862238-01-4

A novel potent, selective Sirt2 inhibitor with IC50 of 0.118 uM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 963 Get Quote
50MG 1962 Get Quote
100MG 2520 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    MZ-242
  • Note
    Research use only, not for human use.
  • Brief Description
    A novel potent, selective Sirt2 inhibitor with IC50 of 0.118 uM.
  • Description
    A novel potent, selective Sirt2 inhibitor with IC50 of 0.118 uM; displays no inhibitory activity against Sirt1 and Sirt 3 (IC50>100 uM).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    MZ242 | MZ242
  • Pathway
    Chromatin/Epigenetic
  • Target
    Sirtuin
  • Recptor
    Sirtuin
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1862238-01-4
  • Formula Weight
    525.646
  • Molecular Formula
    C24H27N7O3S2
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    O=C(NC1=NC=C(CC2=CC=CC(OCC3=CN(CCOC)N=N3)=C2)S1)CSC4=NC(C)=CC(C)=N4
  • Chemical Name
    2-((4,6-dimethylpyrimidin-2-yl)thio)-N-(5-(3-((1-(2-methoxyethyl)-1H-1,2,3-triazol-4-yl)methoxy)benzyl)thiazol-2-yl)acetamide

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Szabó A, et al. Sci Rep. 2017 Dec 6;7(1):17070. 2. Schiedel M, et al. Angew Chem Int Ed Engl. 2016 Feb 5;55(6):2252-6.
molnova catalog
related products
  • lithospermic acid B

    lithospermic acid B is a water-soluble antioxidant from Salvia extract. It plays significant role of antioxidant effect; antiplatelet aggregation anticoagulant and antithrombotic effect.

  • OSS-128167

    OSS-128167 is a novel selective, cell permeable SIRT6 inhibitor.

  • E1231

    E1231 (E-1231) is a small molecule SIRT1 activator with EC50 of 0.83 uM.