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Lartesertib
CAS No. 2495096-26-7
Lartesertib( —— )
Catalog No. M35661 CAS No. 2495096-26-7
Lartesertib (ATM Inhibitor-5) is an inhibitor of serine/threonine protein kinase ATM with potential anticancer activity for the study of lung cancer.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 201 | Get Quote |
|
| 5MG | 312 | Get Quote |
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| 10MG | 534 | Get Quote |
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| 25MG | 1003 | Get Quote |
|
| 50MG | 1674 | Get Quote |
|
| 100MG | 2538 | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameLartesertib
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NoteResearch use only, not for human use.
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Brief DescriptionLartesertib (ATM Inhibitor-5) is an inhibitor of serine/threonine protein kinase ATM with potential anticancer activity for the study of lung cancer.
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DescriptionLartesertib (M4076) is a potent inhibitor of serine/threonine protein kinase ATM (extracted from patent WO2022058351A1).
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayCell Cycle/DNA Damage
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TargetATM/ATR
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RecptorATM/ATR
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Research Area——
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Indication——
Chemical Information
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CAS Number2495096-26-7
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Formula Weight448.45
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Molecular FormulaC23H21FN6O3
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : ≥ 100 mg/mL (222.99 mM)
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SMILESCOc1cncc(F)c1-n1c2c(cnc3cc(OC)c(cc23)-c2cn(C)nc2C)n(C)c1=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Alessandra AMBRUOSI, et al. Pharmaceutical preparation. WO2022058351A1.
molnova catalog
related products
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KU-60019 (b)
KU-60019 is an improved analogue of KU-55933, with IC50 of 6.3 nM for ATM in cell-free assays.
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KU-55933
KU-55933 is a potent, specific, ATP-competitive inhibitor of ATM with Ki/IC50 of 2.2/13 nM.
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KU-60019
KU-60019 is an improved analogue of KU-55933, and is a potent, specific inhibitor of ATM kinase with IC50 of 6.3 nM, 270- and 1,600-fold selectivity over DNA-PKcs and ATR.
