HIF-2α-IN-2

CAS No. 1672666-82-8

HIF-2α-IN-2( —— )

Catalog No. M23751 CAS No. 1672666-82-8

HIF-2α-IN-2 is a hypoxia-inducible factor (HIF-2α) inhibitor (IC50: 16 nM in scintillation proximity assay).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    HIF-2α-IN-2
  • Note
    Research use only, not for human use.
  • Brief Description
    HIF-2α-IN-2 is a hypoxia-inducible factor (HIF-2α) inhibitor (IC50: 16 nM in scintillation proximity assay).
  • Description
    HIF-2α-IN-2 is a hypoxia-inducible factor (HIF-2α) inhibitor (IC50: 16 nM in scintillation proximity assay).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Angiogenesis
  • Target
    HIF/HIF Prolyl-hydroxylase
  • Recptor
    HIF-2α
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1672666-82-8
  • Formula Weight
    365.35
  • Molecular Formula
    C17H13F2NO4S
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:100 mg/mL (273.71 mM; Need ultrasonic)
  • SMILES
    N#CC1=CC(OC2=CC=C(S(=O)(C)=O)C3=C2CC(F)C3O)=CC(F)=C1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Darryl David DIXON, et al. Aryl ethers and uses thereof. WO2015035223A1.
molnova catalog
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