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Endoxifen
CAS No. 112093-28-4
Endoxifen( —— )
Catalog No. M10432 CAS No. 112093-28-4
A metabolite of tamoxifen, orally active non-steroidal selective estrogen receptor modulator (SERM) for the treatment of estrogen receptor-positive breast cancer.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 73 | In Stock |
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| 5MG | 120 | In Stock |
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| 10MG | 192 | In Stock |
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| 25MG | 356 | In Stock |
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| 50MG | 555 | In Stock |
|
| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameEndoxifen
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NoteResearch use only, not for human use.
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Brief DescriptionA metabolite of tamoxifen, orally active non-steroidal selective estrogen receptor modulator (SERM) for the treatment of estrogen receptor-positive breast cancer.
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DescriptionA metabolite of tamoxifen, orally active non-steroidal selective estrogen receptor modulator (SERM) for the treatment of estrogen receptor-positive breast cancer.Breast Cancer Phase 1 Clinical.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayEndocrinology/Hormones
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TargetEstrogen Receptor/ERR
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RecptorER|ERR|hERGPotassiumChannel
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Research AreaCancer
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IndicationBreast Cancer
Chemical Information
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CAS Number112093-28-4
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Formula Weight373.4874
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Molecular FormulaC25H27NO2
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Purity>98% (HPLC)
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Solubility10 mM in DMSO
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SMILESCCC(=C(C1=CC=C(C=C1)O)C2=CC=C(C=C2)OCCNC)C3=CC=CC=C3
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Chemical NamePhenol, 4-[(1Z)-1-[4-[2-(methylamino)ethoxy]phenyl]-2-phenyl-1-buten-1-yl]-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Brauch H, et al. Clin Chem. 2009 Oct;55(10):1770-82.
2. Markopoulos C, et al. World J Clin Oncol. 2014 Aug 10;5(3):374-81.
3. Mugundu GM, et al. Drug Metab Dispos. 2012 Feb;40(2):389-96.
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