CTAP(TFA）( —— )

Catalog No. M22905 CAS No. ——

COA

Datasheet

HNMR

HPLC

MSDS

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Product Name

CTAP(TFA）
Note

Research use only, not for human use.
Brief Description

CTAP TFA is a potent, highly selective, and brain penetrant antagonist of μ-opioid receptor with IC50 of 3.5 nM. It displays over 1200-fold selectivity over δ opioid (IC50=4500 nM) and somatostatin receptors.
Description

CTAP TFA is a potent, highly selective, and brain penetrant antagonist of μ-opioid receptor with IC50 of 3.5 nM. It displays over 1200-fold selectivity over δ opioid (IC50=4500 nM) and somatostatin receptors. CTAP TFA can be used for the study of L-DOPA-induced dyskinesia (LID).
In Vitro

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In Vivo

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Synonyms

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Pathway

Endocrinology/Hormones
Target

Opioid Receptor
Recptor

δ-opioid receptor
Research Area

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Indication

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CAS Number

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Formula Weight

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Molecular Formula

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Purity

>98% (HPLC)
Solubility

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SMILES

CC(O)C1C(NC(C(NC(C(N)=O)C(O)C)=O)C(C)(C)SSCC(NC(C(N)CC2=CC=CC=C2)=O)C(NC(CC3=CC=C(O)C=C3)C(NC(CC4=CNC5=CC=CC=C54)C(NC(CCC/N=C(N)\N)C(N1)=O)=O)=O)=O)=O.O=C(O)C(F)(F)F
Chemical Name

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1.Mitchell J Bartlett, et al. Highly-selective μ-opioid Receptor Antagonism Does Not Block L-DOPA-induced Dyskinesia in a Rodent Model.BMC Res Notes

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