Deltorphin 2(TFA)

CAS No. 122752-16-3

Deltorphin 2(TFA)( [D-Ala2]-Deltorphin II )

Catalog No. M21044 CAS No. 122752-16-3

Deltorphin 2(TFA) is an agonist of δ opioid receptor(IC50:0.41 nM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 168 In Stock
10MG 311 In Stock
25MG 527 In Stock
50MG 742 In Stock
100MG 1014 In Stock
200MG Get Quote In Stock
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Biological Information

  • Product Name
    Deltorphin 2(TFA)
  • Note
    Research use only, not for human use.
  • Brief Description
    Deltorphin 2(TFA) is an agonist of δ opioid receptor(IC50:0.41 nM).
  • Description
    Deltorphin 2(TFA) is an agonist of δ opioid receptor(IC50:0.41 nM).
  • In Vitro
    Deltorphin 2 ([D-Ala2]-Deltorphin II) is enzymatically stable, amphibian heptapeptides that has a high affinity and selectivity for delta-opioid receptor. Deltorphin 2 is the most selective natural delta opioid receptor agonist.
  • In Vivo
    ——
  • Synonyms
    [D-Ala2]-Deltorphin II
  • Pathway
    Endocrinology/Hormones
  • Target
    Opioid Receptor
  • Recptor
    δ-opioid receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    122752-16-3
  • Formula Weight
    782.88
  • Molecular Formula
    C38H54N8O10
  • Purity
    >98% (HPLC)
  • Solubility
    H2O:7.5 mg/mL (9.58 mM; Need ultrasonic and warming)
  • SMILES
    CC(C)[C@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@H](C(=O)NCC(N)=O)C(C)C
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Thomas S A Abbruscato T J Hau V S et al. Structure-Activity Relationships of a Series of [D-Ala2]Deltorphin I and II Analogues ;[J]. Journal of Pharmacology and Experimental Therapeutics 1997 281(2):817-825.
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