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Deltorphin 2(TFA)
CAS No. 122752-16-3
Deltorphin 2(TFA)( [D-Ala2]-Deltorphin II )
Catalog No. M21044 CAS No. 122752-16-3
Deltorphin 2(TFA) is an agonist of δ opioid receptor(IC50:0.41 nM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 159 | Get Quote |
|
| 10MG | 294 | Get Quote |
|
| 25MG | 500 | Get Quote |
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| 50MG | 718 | Get Quote |
|
| 100MG | 981 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameDeltorphin 2(TFA)
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NoteResearch use only, not for human use.
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Brief DescriptionDeltorphin 2(TFA) is an agonist of δ opioid receptor(IC50:0.41 nM).
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DescriptionDeltorphin 2(TFA) is an agonist of δ opioid receptor(IC50:0.41 nM).
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In VitroDeltorphin 2 ([D-Ala2]-Deltorphin II) is enzymatically stable, amphibian heptapeptides that has a high affinity and selectivity for delta-opioid receptor. Deltorphin 2 is the most selective natural delta opioid receptor agonist.
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In Vivo——
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Synonyms[D-Ala2]-Deltorphin II
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PathwayEndocrinology/Hormones
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TargetOpioid Receptor
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Recptorδ-opioid receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number122752-16-3
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Formula Weight782.88
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Molecular FormulaC38H54N8O10
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Purity>98% (HPLC)
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SolubilityH2O:7.5 mg/mL (9.58 mM; Need ultrasonic and warming)
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SMILESCC(C)[C@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@H](C(=O)NCC(N)=O)C(C)C
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Thomas S A Abbruscato T J Hau V S et al. Structure-Activity Relationships of a Series of [D-Ala2]Deltorphin I and II Analogues ;[J]. Journal of Pharmacology and Experimental Therapeutics 1997 281(2):817-825.
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