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Bremelanotide
CAS No. 189691-06-3
Bremelanotide( PT-141 | PT 141 )
Catalog No. M12979 CAS No. 189691-06-3
A peptide, non-selective melanocortin receptor agonist for treatment for female sexual dysfunction.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 100MG | Get Quote | In Stock |
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| 200MG | Get Quote | In Stock |
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| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
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Biological Information
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Product NameBremelanotide
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NoteResearch use only, not for human use.
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Brief DescriptionA peptide, non-selective melanocortin receptor agonist for treatment for female sexual dysfunction.
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DescriptionA peptide, non-selective melanocortin receptor agonist for treatment for female sexual dysfunction; selectively stimulates solicitational behaviors in the female rat, without affecting lordosis, pacing, or other sexual behaviors, does not cause generalized motor activation; a peptide analogue of α-MSH.Sexual Dysfunction Phase 3 Clinical.
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In Vitro——
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In Vivo——
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SynonymsPT-141 | PT 141
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PathwayGPCR/G Protein
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TargetMelanocortin Receptor
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RecptorMelanocortin Receptor
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Research AreaEndocrinology
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IndicationSexual Dysfunction
Chemical Information
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CAS Number189691-06-3
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Formula Weight1025.2
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Molecular FormulaC50H68N14O10
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Purity>98% (HPLC)
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Solubility——
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SMILESCCCCC(C(=O)NC1CC(=O)NCCCCC(NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC1=O)CC2=CN=CN2)CC3=CC=CC=C3)CCCN=C(N)N)CC4=CNC5=CC=CC=C54)C(=O)O)NC(=O)C
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Chemical NameN-Acetyl-L-norleucyl-L-alpha-aspartyl-L-histidyl-D-phenylalanyl-L-arginyl-L-tryptophyl-L-lysine (2-7)-lactam
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Pfaus JG, et al. Proc Natl Acad Sci U S A. 2004 Jul 6;101(27):10201-4.
2. Molinoff PB, et al. Ann N Y Acad Sci. 2003 Jun;994:96-102.
3. Aughton KL, et al.
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