Cart
sales@molnova.com
Home - Products - Endocrinology/Hormones - Opioid Receptor - AT-121

AT-121

CAS No. 2099681-31-7

AT-121( —— )

Catalog No. M34966 CAS No. 2099681-31-7

AT-121 is a dual μ-opioid and neuropeptide receptor partial agonist (Kis 16.49 and 3.67 nM, respectively).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 532 Get Quote
5MG 787 Get Quote
10MG 1074 Get Quote
25MG 1463 Get Quote
50MG 1822 Get Quote
100MG 2250 Get Quote
500MG 4410 Get Quote
1G Get Quote Get Quote
Get Quotation Bulk Inquiry Add to Cart

Biological Information

  • Product Name
    AT-121
  • Note
    Research use only, not for human use.
  • Brief Description
    AT-121 is a dual μ-opioid and neuropeptide receptor partial agonist (Kis 16.49 and 3.67 nM, respectively).
  • Description
    AT-121 is a bifunctional nociception and mu opioid receptor agonist, with Kis of 3.67 and 16.49 nM, respectively. AT-121 is a safe, non-addictive analgesic, and shows antinociceptive and antiallodynic effects.
  • In Vitro
    ——
  • In Vivo
    AT-121 (0.003-0.03 mg/kg; s.c.) produces potent antinociceptive effect.Animal Model:Adult male and female rhesus monkeysDosage:0.003-0.03 mg/kg Administration:Subcutaneous Result:Produced antinociceptive effects against an acute noxious stimulus, 50 °C water, in a dose-dependent.
  • Synonyms
    ——
  • Pathway
    Endocrinology/Hormones
  • Target
    Opioid Receptor
  • Recptor
    Opioid Receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2099681-31-7
  • Formula Weight
    462.65
  • Molecular Formula
    C24H38N4O3S
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    O=C1C2(C=3C(CN1CCNS(N)(=O)=O)=CC=CC3)CCN(CC2)[C@@H]4CC[C@H]([C@H](C)C)CC4
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Ding H, Kiguchi N, Yasuda D, et al. A bifunctional nociceptin and mu opioid receptor agonist is analgesic without opioid side effects in nonhuman primates. Sci Transl Med. 2018;10(456):eaar3483. doi:10.1126/scitranslmed.aar3483?
Calculator

Molecular Weight Calculator

Dilution Calculator

Molarity Calculator

molnova catalog
related products

  • Salvinorin A

    Salvinorin A is a non-nitrogenous κ-opioid selective agonist.

  • SCH 486757

    A novel potent, selective, orally active nociceptin/orphanin FQ peptide (NOP, ORL1) receptor agonist with Ki of 4.6 nM, with high selectiivity over classical opioid receptors.

  • CP 866087

    CP 866087 is an opioid receptor antagonist for the study of female sexual dysfunction.

Sign In Join Free