
SAR407899 hydrochloride
SAR407899 hydrochloride
Catalog No. M27702
SAR407899 hydrochloride is a selective, potent and ATP-competitive ROCK inhibitor, with an IC50 of 135 nM for ROCK-2, and Kis of 36 nM and 41 nM for human and rat ROCK-2, respectively.
Size | Price / USD | Stock | Quantity |
5MG | 42 | Get Quote |
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10MG | 65 | Get Quote |
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25MG | 115 | Get Quote |
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50MG | 200 | Get Quote |
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100MG | 320 | Get Quote |
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500MG | 758 | Get Quote |
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1G | Get Quote | Get Quote |
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Biological Information
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Product NameSAR407899 hydrochloride
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Brief Description
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Description
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Storage
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NoteResearch use only, not for human use.
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Reference1.Ford AP, et al. RS-17053 (N-[2-(2-cyclopropylmethoxyphenoxy)ethyl]-5-chloro-alpha, alpha-dimethyl-1H-indole-3-ethanamine hydrochloride), a selective alpha 1A-adrenoceptor antagonist, displays low affinity for functional alpha 1-adrenoceptors in human prostate: implications for adrenoceptor classification. Mol Pharmacol. 1996 Feb;49(2):209-15.
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