SAR407899 hydrochloride

SAR407899 hydrochloride

Catalog No. M27702

SAR407899 hydrochloride is a selective, potent and ATP-competitive ROCK inhibitor, with an IC50 of 135 nM for ROCK-2, and Kis of 36 nM and 41 nM for human and rat ROCK-2, respectively.

Size Price / USD Stock Quantity
5MG 42 Get Quote
10MG 65 Get Quote
25MG 115 Get Quote
50MG 200 Get Quote
100MG 320 Get Quote
500MG 758 Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    SAR407899 hydrochloride
  • Brief Description
  • Description
  • Storage
  • Note
    Research use only, not for human use.
  • Reference
    1.Ford AP, et al. RS-17053 (N-[2-(2-cyclopropylmethoxyphenoxy)ethyl]-5-chloro-alpha, alpha-dimethyl-1H-indole-3-ethanamine hydrochloride), a selective alpha 1A-adrenoceptor antagonist, displays low affinity for functional alpha 1-adrenoceptors in human prostate: implications for adrenoceptor classification. Mol Pharmacol. 1996 Feb;49(2):209-15.
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