
AM095 free acid
AM095 free acid
Catalog No. M22924
AM095 (free acid) is a potent LPA1 receptor antagonist (IC50s: 0.98 and 0.73 μM for recombinant human or mouse LPA1).In vitro, AM095 was a potent LPA receptor antagonist because it inhibited GTPγS binding to Chinese hamster ovary (CHO) cell membranes overexpressing recombinant human or mouse LPA with IC values of 0.98 and 0.73 μM, respectively, and exhibited no LPA agonism.
Size | Price / USD | Stock | Quantity |
2MG | 42 | In Stock |
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5MG | 68 | In Stock |
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10MG | 110 | In Stock |
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25MG | 200 | In Stock |
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50MG | 335 | In Stock |
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100MG | 520 | In Stock |
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200MG | 750 | In Stock |
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500MG | Get Quote | In Stock |
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1G | Get Quote | In Stock |
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Biological Information
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Product NameAM095 free acid
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Brief Description
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Description
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Storage
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NoteResearch use only, not for human use.
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Reference1. Castelino FV, et al. Amelioration of dermal fibrosis by genetic deletion or pharmacologic antagonism of lysophosphatidic acid receptor 1 in a mouse model of scleroderma. Arthritis Rheum. 2011 May;63(5):1405-15.
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