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Tezampanel

CAS No. 150131-78-5

Tezampanel( LY 293558 | NGX 424 )

Catalog No. M12089 CAS No. 150131-78-5

Tezampanel (LY 293558, NGX 424) is a competitive antagonist of the AMPA and kainate receptors with selectivity for the GluR5 subtype of the kainate receptor.

Purity : >98% (HPLC)

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Biological Information

  • Product Name
    Tezampanel
  • Note
    Research use only, not for human use.
  • Brief Description
    Tezampanel (LY 293558, NGX 424) is a competitive antagonist of the AMPA and kainate receptors with selectivity for the GluR5 subtype of the kainate receptor.
  • Description
    Tezampanel (LY 293558, NGX 424) is a competitive antagonist of the AMPA and kainate receptors with selectivity for the GluR5 subtype of the kainate receptor; has neuroprotective and anticonvulsant properties, also has anxiolytic effects in animal studies.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    LY 293558 | NGX 424
  • Pathway
    Membrane Transporter/Ion Channel
  • Target
    iGluR
  • Recptor
    iGluR
  • Research Area
    Neurological Disease
  • Indication
    Migraine

Chemical Information

  • CAS Number
    150131-78-5
  • Formula Weight
    279.344
  • Molecular Formula
    C13H21N5O2
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    C1CC2CNC(CC2CC1CCC3=NNN=N3)C(=O)O
  • Chemical Name
    (3S,4aR,6R,8aR)-6-[2-(1H-tetrazol-5-yl)ethyl]decahydroisoquinoline-3-carboxylic acid

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Ornstein PL, et al. J Med Chem. 1993 Jul 9;36(14):2046-8. 2. LeBlanc MH, et al. Stroke. 1995 Oct;26(10):1908-14; discussion 1914-5. 3. Benvenga MJ, et al. J Pharmacol Exp Ther. 1995 Oct;275(1):164-70.
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