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Obicetrapib
CAS No. 866399-87-3
Obicetrapib( AMG-899 | AMG899 | TA-8995 | DEX-001 )
Catalog No. M16296 CAS No. 866399-87-3
Obicetrapib (AMG-899, TA-8995, DEX-001) is a potent, ora cholesteryl ester transfer protein (CETP) inhibitor for treatment of dyslipidaemia.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 212 | In Stock |
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| 5MG | 154 | In Stock |
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| 10MG | 216 | In Stock |
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| 25MG | 390 | In Stock |
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| 100MG | Get Quote | In Stock |
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| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameObicetrapib
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NoteResearch use only, not for human use.
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Brief DescriptionObicetrapib (AMG-899, TA-8995, DEX-001) is a potent, ora cholesteryl ester transfer protein (CETP) inhibitor for treatment of dyslipidaemia.
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DescriptionObicetrapib (AMG-899, TA-8995, DEX-001) is a potent, ora cholesteryl ester transfer protein (CETP) inhibitor for treatment of dyslipidaemia.Dyslipidemia Phase 2 Clinical.
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In Vitro——
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In Vivo——
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SynonymsAMG-899 | AMG899 | TA-8995 | DEX-001
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PathwayMetabolic Enzyme/Protease
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TargetCETP
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RecptorCETP
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Research AreaCardiovascular Disease
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IndicationDyslipidemia
Chemical Information
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CAS Number866399-87-3
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Formula Weight722.609
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Molecular FormulaC32H31F9N4O5
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Purity>98% (HPLC)
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Solubility——
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SMILESCCC1CC(C2=C(N1C(=O)OCC)C=CC(=C2)C(F)(F)F)N(CC3=CC(=CC(=C3)C(F)(F)F)C(F)(F)F)C4=NC=C(C=N4)OCCCC(=O)O
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Chemical Name4-[2-[[3,5-bis(trifluoromethyl)phenyl]methyl-[(2R,4S)-1-ethoxycarbonyl-2-ethyl-6-(trifluoromethyl)-3,4-dihydro-2H-quinolin-4-yl]amino]pyrimidin-5-yl]oxybutanoic acid
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Ford J, et al. Br J Clin Pharmacol. 2014 Sep;78(3):498-508.
2. Hovingh GK, et al. Lancet. 2015 Aug 1;386(9992):452-60.
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