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Maropitant
CAS No. 147116-67-4
Maropitant( —— )
Catalog No. M20648 CAS No. 147116-67-4
Maropitant is a selective neurokinin (NK1) receptor antagonist.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 39 | In Stock |
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| 5MG | 65 | In Stock |
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| 10MG | 110 | In Stock |
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| 25MG | 177 | In Stock |
|
| 50MG | 335 | In Stock |
|
| 100MG | 500 | In Stock |
|
| 500MG | 1098 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameMaropitant
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NoteResearch use only, not for human use.
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Brief DescriptionMaropitant is a selective neurokinin (NK1) receptor antagonist.
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DescriptionMaropitant is a selective neurokinin (NK1) receptor antagonist.
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In Vitro——
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In VivoTreatment with 1 mg/kg Maropitant citrate, significantly reduces the size of ulcerative dermatitis (UD) lesions in mice. Intravenous Maropitant decreases MAC by 16%. In contrast, epidural administration of either saline or Maropitant does not change the MAC (2.17% and 1.92 %, respectively).
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Synonyms——
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PathwayGPCR/G Protein
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TargetNeurokinin Receptor
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RecptorNK1
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Research Area——
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Indication——
Chemical Information
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CAS Number147116-67-4
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Formula Weight468.67
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Molecular FormulaC32H40N2O
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Purity>98% (HPLC)
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SolubilityDMSO:33.33 mg/mL (71.12 mM)
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SMILESCOc1ccc(cc1CN[C@H]1C2CCN(CC2)[C@H]1C(c1ccccc1)c1ccccc1)C(C)(C)C
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Hickman M A Cox S R Mahabir S et al. Safety pharmacokinetics and use of the novel NK‐1 receptor antagonist maropitant (Cerenia TM ) for the prevention of emesis and motion sickness in cats[J]. Journal of Veterinary Pharmacology and Therapeutics 2008 31(3):220-229.
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