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Burapitant
CAS No. 537034-22-3
Burapitant( —— )
Catalog No. M36273 CAS No. 537034-22-3
Burapitant (SSR 240600) is a novel non-peptide tachykinin neurokinin 1 (NK) receptor antagonist with anti-coke oven and antidepressant activity.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 1502 | Get Quote |
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| 5MG | 1881 | Get Quote |
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| 25MG | 2640 | Get Quote |
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| 50MG | 3110 | Get Quote |
|
| 100MG | 4140 | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameBurapitant
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NoteResearch use only, not for human use.
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Brief DescriptionBurapitant (SSR 240600) is a novel non-peptide tachykinin neurokinin 1 (NK) receptor antagonist with anti-coke oven and antidepressant activity.
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DescriptionBurapitant (SSR 240600) is a novel non-peptide tachykinin neurokinin 1 (NK) receptor antagonist with anti-coke oven and antidepressant activity.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayGPCR/G Protein
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TargetNeurokinin Receptor
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RecptorNeurokinin receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number537034-22-3
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Formula Weight682.52
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Molecular FormulaC31H35Cl2F6N3O3
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Purity>98% (HPLC)
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Solubility——
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SMILESC(CN1CCC(C(C(N)=O)(C)C)CC1)[C@]2(CN(C(CC3=CC(C(F)(F)F)=CC(C(F)(F)F)=C3)=O)CCO2)C4=CC(Cl)=C(Cl)C=C4
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
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Rolapitant hydrochlo...
Rolapitant (SCH619734) hydrochloride is a potent, selective, long-acting, and orally active neurokinin 1 (NK1) receptor antagonist with a K_i of 0.66 nM, which does not interact with CYP3A4 and demonstrates potent centrally-mediated anti-emetic activity in both acute and delayed ferret emesis models .
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Talnetant
Talnetant is a selective competitive brain-penetrant NK3 receptor antagonist with the ability to modulate mesolimbic and mesocortical dopaminergic neurotransmission.
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Eledoisin
Eledoisin is a specific agonist of NK2 and NK3 receptors.Eledoisin is an undecapeptide of mollusk origin, belonging to the tachykinin family of neuropeptides.Eledoisin increases the value recorded under basal conditions by 24.5±3.7%; this stimulation is significantly (P<0.01) lowered to 13.1±1.9% by the simultaneous presence of CP99994.
