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MK-204
CAS No. 1959605-73-2
MK-204( MK204 )
Catalog No. M13074 CAS No. 1959605-73-2
MK-204 is a potent, selective AKR1B10 inhibitor with IC50 of 80 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 873 | Get Quote |
|
| 50MG | 1782 | Get Quote |
|
| 100MG | 2250 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
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Biological Information
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Product NameMK-204
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NoteResearch use only, not for human use.
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Brief DescriptionMK-204 is a potent, selective AKR1B10 inhibitor with IC50 of 80 nM.
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DescriptionMK-204 is a potent, selective AKR1B10 inhibitor with IC50 of 80 nM, shows high selective (270-fold) over AKR1B1; a lead compound targeting the distinct AKR1B10 specificity pocket and with a strong X-bond.
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In Vitro——
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In Vivo——
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SynonymsMK204
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PathwayMetabolic Enzyme/Protease
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TargetAldose Reductase
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RecptorAldose Reductase
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Research Area——
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Indication——
Chemical Information
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CAS Number1959605-73-2
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Formula Weight714.221
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Molecular FormulaC16H9Br5ClNO4
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Purity>98% (HPLC)
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Solubility——
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SMILESO=C(O)COC1=CC(Cl)=CC=C1C(NCC2=C(Br)C(Br)=C(Br)C(Br)=C2Br)=O
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Chemical NameAcetic acid, 2-[5-chloro-2-[[[(2,3,4,5,6-pentabromophenyl)methyl]amino]carbonyl]phenoxy]-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Cousido-Siah A, et al. ACS Chem Biol. 2016 Oct 21;11(10):2693-2705.
molnova catalog
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