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Endothelin-1 (11-21)
CAS No. 144602-02-8
Endothelin-1 (11-21)( ——— )
Catalog No. M41119 CAS No. 144602-02-8
IRL 1038 is an endothelin B receptor selective antagonist with a Ki of 6-11 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
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Biological Information
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Product NameEndothelin-1 (11-21)
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NoteResearch use only, not for human use.
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Brief DescriptionIRL 1038 is an endothelin B receptor selective antagonist with a Ki of 6-11 nM.
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DescriptionETB endothelin receptor antagonist
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In Vitro———
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In Vivo———
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Synonyms———
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PathwayGPCR/G Protein
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TargetEndothelin Receptor
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RecptorETB endothelin receptor
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Research Area———
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Indication———
Chemical Information
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CAS Number144602-02-8
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Formula Weight1409.67
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Molecular FormulaC68H92N14O15S2
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Purity>98% (HPLC)
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Solubility———
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SMILES———
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Urade Y, et al. An endothelin B receptor-selective antagonist: IRL 1038, Cys11-Cys15-endothelin-1(11-21). FEBS Lett. 1992 Oct 12;311(1):12-6. doi: 10.1016/0014-5793(92)81355-p.?
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