[Ala1,3,11,15]-Endothelin

Research use only, not for human use.

Selective ETB endothelin receptor agonist (IC50 values are 0.33 and 2200 nM for displacing [125I]-ET-1 from ETB and ETA receptors respectively).

Selective ETB endothelin receptor agonist (IC50 values are 0.33 and 2200 nM for displacing [125I]-ET-1 from ETB and ETA receptors respectively).

[Ala1,3,11,15]-Endothelin (53-63) (0.1 μM) has selectivity for ETB with IC50 values of 0.61 nM, 0.61 nM, 0.33 nM, 2200 nM in Bronchus, Lung, Cerebellum and VSMC, respectively.

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GPCR/G Protein

Endothelin Receptor

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121204-87-3

2368

C109H163N25O32S

>98% (HPLC)

water:1 mg/mL

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(-20℃)

With Ice Pack

≥ 2 years