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Acetyl-(Ala11·15)-Endothelin-1 (6-21)
CAS No. 143113-45-5
Acetyl-(Ala11·15)-Endothelin-1 (6-21)( ——— )
Catalog No. M40168 CAS No. 143113-45-5
BQ-3020 is a selective endothelin receptor (ETB receptor) agonist that displaces [125I] ET-1 binding to ETB receptors, with an IC50 value of 0.2 nM. BQ-3020 elicits vasoconstriction in the rabbit pulmonary artery. BQ-3020 makes relaxation of the pig urinary bladder neck and can be used for cardiovascular disease research12.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
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Biological Information
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Product NameAcetyl-(Ala11·15)-Endothelin-1 (6-21)
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NoteResearch use only, not for human use.
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Brief DescriptionBQ-3020 is a selective endothelin receptor (ETB receptor) agonist that displaces [125I] ET-1 binding to ETB receptors, with an IC50 value of 0.2 nM. BQ-3020 elicits vasoconstriction in the rabbit pulmonary artery. BQ-3020 makes relaxation of the pig urinary bladder neck and can be used for cardiovascular disease research12.
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DescriptionBQ-3020 is a selective endothelin receptor (ETB receptor) agonist that displaces [125I] ET-1 binding to ETB receptors, with an IC50 value of 0.2 nM.
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In Vitro———
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In VivoAnimal Model:Cancer pain mouse model Dosage:3 mg/kg Administration:Injected subcutaneously at the site of the greatest tumor development Result:Attenuated cancer pain by approximately 50% up to 3 h post-injection compared to PBS-vehicle and contralateral injection
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Synonyms———
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PathwayOthers
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TargetOther Targets
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RecptorETB: 0.2 nM (IC50)
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Research Area———
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Indication———
Chemical Information
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CAS Number143113-45-5
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Formula Weight1989.36
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Molecular FormulaC96H139N20O24S
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Purity>98% (HPLC)
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Solubility———
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SMILES———
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Arteaga JL,et.al. Endothelin ET(B) receptors are involved in the relaxation to the pig urinary bladder neck. Neurourol Urodyn. 2012 Jun;31(5):688-94. ?
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