EZH2-IN-2

CAS No. 2238821-31-1

EZH2-IN-2( ——— )

Catalog No. M39456 CAS No. 2238821-31-1

EZH2-IN-2 is a EZH2 inhibitor extracted from patent WO2018133795A1, Compound Example 69, with an IC50 of 64 nM. EZH2-IN-2 can be used for the research of cancer or precancerous condition related to EZH2 activity.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    EZH2-IN-2
  • Note
    Research use only, not for human use.
  • Brief Description
    EZH2-IN-2 is a EZH2 inhibitor extracted from patent WO2018133795A1, Compound Example 69, with an IC50 of 64 nM. EZH2-IN-2 can be used for the research of cancer or precancerous condition related to EZH2 activity.
  • Description
    EZH2-IN-2 is a EZH2 inhibitor extracted from patent WO2018133795A1, Compound Example 69, with an IC50 of 64 nM.
  • In Vitro
    ———
  • In Vivo
    ———
  • Synonyms
    ———
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    EZH2: 64 nM (IC50)
  • Research Area
    ———
  • Indication
    ———

Chemical Information

  • CAS Number
    2238821-31-1
  • Formula Weight
    610.79
  • Molecular Formula
    C36H46N6O3
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO : 10 mg/mL (16.37 mM; ultraphonic (<60°C); )
  • SMILES
    ———
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. LIU, Qing Song, et al. Ezh2 inhibitor and use thereof. WO2018133795A1.
molnova catalog
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