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KSK68
CAS No. 2566715-91-9
KSK68( —— )
Catalog No. M37239 CAS No. 2566715-91-9
KSK68 is a potent dual sigma-1 and histamine H3 receptor antagonist with potential analgesic activity and high affinity for H3 receptors, sigma-1, sigma-2 receptors.KSK68 can be used in the study of pain related diseases.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 103 | Get Quote |
|
| 5MG | 155 | Get Quote |
|
| 10MG | 226 | Get Quote |
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| 25MG | 363 | Get Quote |
|
| 50MG | 546 | Get Quote |
|
| 100MG | 761 | Get Quote |
|
| 500MG | 2115 | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameKSK68
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NoteResearch use only, not for human use.
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Brief DescriptionKSK68 is a potent dual sigma-1 and histamine H3 receptor antagonist with potential analgesic activity and high affinity for H3 receptors, sigma-1, sigma-2 receptors.KSK68 can be used in the study of pain related diseases.
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DescriptionKSK68 is a high-affinity dual sigma-1 and histamine H3 receptor antagonist, with Kis of 7.7, 3.6, 22.4 nM for H3 receptor, sigma-1, sigma-2 receptor respectively. KSK68 has negligible affinity at the other histamine receptor subtypes. KSK68 can be used for research of nociceptive and neuropathic pain.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayGPCR/G Protein
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TargetHistamine Receptor
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RecptorHistamine Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number2566715-91-9
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Formula Weight364.48
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Molecular FormulaC23H28N2O2
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Purity>98% (HPLC)
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Solubility——
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SMILESO=C(C1=CC=C(OCCCN2CCC(C=3C=CN=CC3)CC2)C=C1)C4CC4
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Szczepańska K, et al. Dual Piperidine-Based Histamine H3 and Sigma-1 Receptor Ligands in the Treatment of Nociceptive and Neuropathic Pain. J Med Chem. 2023 Jul 27;66(14):9658-9683.?
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