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ERK5-IN-6
CAS No. 2734916-64-2
ERK5-IN-6( —— )
Catalog No. M37089 CAS No. 2734916-64-2
ERK5-IN-6 is a potent inhibitor of ERK5 kinase.ERK5-IN-6 exhibits antiproliferative activity, anticonvulsant activity, and antitumor activity, and can be used in the study of central nervous system-related disorders.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 296 | In Stock |
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| 5MG | 459 | In Stock |
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| 10MG | 657 | In Stock |
|
| 25MG | 994 | In Stock |
|
| 50MG | 1371 | In Stock |
|
| 100MG | 1773 | In Stock |
|
| 500MG | 3537 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameERK5-IN-6
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NoteResearch use only, not for human use.
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Brief DescriptionERK5-IN-6 is a potent inhibitor of ERK5 kinase.ERK5-IN-6 exhibits antiproliferative activity, anticonvulsant activity, and antitumor activity, and can be used in the study of central nervous system-related disorders.
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DescriptionERK5-IN-6 (compound 5J)is an ERK5 kinase inhibitor with anticancer activity. ERK5-IN-6 exhibits good anti-proliferative activity with the IC50 value of 4.56 μg/mL for A549 cells.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayMAPK/ERK Signaling
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TargetERK
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RecptorERK
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Research Area——
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Indication——
Chemical Information
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CAS Number2734916-64-2
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Formula Weight339.43
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Molecular FormulaC23H21N3
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Purity>98% (HPLC)
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Solubility——
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SMILESN1=CC=CC2=C1NC=C2C3=CCN(CC=4C=CC=5C=CC=CC5C4)CC3
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Qin Zhang, et al. Design, synthesis and SAR of novel 7-azaindole derivatives as potential Erk5 kinase inhibitor with anticancer activity. Bioorg Med Chem. 2023 Oct 14:95:117503. ?
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