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PI5P4Ks-IN-2
CAS No. 2766854-03-7
PI5P4Ks-IN-2( —— )
Catalog No. M36403 CAS No. 2766854-03-7
PI5P4Ks-IN-2 is an inhibitor of the phosphatidylinositol 5-phosphate 4-kinase PI5P4Kγ.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 370 | In Stock |
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| 5MG | 337 | In Stock |
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| 10MG | 503 | In Stock |
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| 25MG | 848 | In Stock |
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| 50MG | 1088 | In Stock |
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| 100MG | 1423 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NamePI5P4Ks-IN-2
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NoteResearch use only, not for human use.
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Brief DescriptionPI5P4Ks-IN-2 is an inhibitor of the phosphatidylinositol 5-phosphate 4-kinase PI5P4Kγ.
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DescriptionPI5P4Ks-IN-2 is a inhibitor of phosphatidylinositol 5-phosphate 4-kinase γ (PI5P4Kγ). PI5P4Ks-IN-2 targets to PI5P4K isoforms with pIC50 values of <4.3 (PI5P4Kα), <4.6 (PI5P4Kβ), 6.2 (PI5P4Kγ), 0.32 (PI5P4Kγ+), respectively.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayPI3K/Akt/mTOR signaling
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TargetPI3K
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RecptorPI3K
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Research Area——
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Indication——
Chemical Information
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CAS Number2766854-03-7
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Formula Weight357.45
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Molecular FormulaC22H23N5
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Purity>98% (HPLC)
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Solubility——
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SMILESN(CC1=CC=CC=N1)C2=C3C(=NC(=N2)C4=C(C(C)C)C=CC=C4)C=CN3C
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Boffey HK, et al. Development of Selective Phosphatidylinositol 5-Phosphate 4-Kinase γ Inhibitors with a Non-ATP-competitive, Allosteric Binding Mode. J Med Chem. 2022 Feb 24;65(4):3359-3370. ?
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