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CB2R/FAAH?modulator-1
CAS No. 928892-60-8
CB2R/FAAH?modulator-1( —— )
Catalog No. M36058 CAS No. 928892-60-8
CB2R/FAAH modulator-1, a cannabinoid type 2 receptor (CB2R) agonist, is also a fatty acid amide hydrolase (FAAH) inhibitor (IC50=4 μM) that reduces the production of pro-inflammatory and anti-inflammatory cytokines and is commonly used in inflammation studies.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 110 | In Stock |
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| 5MG | 107 | In Stock |
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| 10MG | 157 | In Stock |
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| 25MG | 236 | In Stock |
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| 50MG | 324 | In Stock |
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| 100MG | 442 | In Stock |
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| 200MG | 594 | In Stock |
|
| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
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Biological Information
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Product NameCB2R/FAAH?modulator-1
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NoteResearch use only, not for human use.
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Brief DescriptionCB2R/FAAH modulator-1, a cannabinoid type 2 receptor (CB2R) agonist, is also a fatty acid amide hydrolase (FAAH) inhibitor (IC50=4 μM) that reduces the production of pro-inflammatory and anti-inflammatory cytokines and is commonly used in inflammation studies.
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DescriptionCB2R/FAAH modulator-1 is a cannabinoid type 2 receptor (CB2R) full agonist with Kis of 14.8 nM and 241.3 nM for CB2R and CB1R, respectively. CB2R/FAAH modulator-1 is a fatty acid amide hydrolase (FAAH) inhibitor with an IC50 of 4 μM. CB2R/FAAH modulator-1 decreases pro-inflammatory and increases anti-inflammatory cytokines production.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayMetabolic Enzyme/Protease
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TargetFAAH
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RecptorFAAH | Cannabinoid Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number928892-60-8
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Formula Weight361.48
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Molecular FormulaC24H27NO2
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Purity>98% (HPLC)
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Solubility——
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SMILESN(C(=O)C1=C(OCC2=CC=CC=C2)C=CC=C1)C34CC5CC(C3)CC(C4)C5
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Francesca Intranuov, et al. Development of N-(1-Adamantyl)benzamides as Novel Anti-Inflammatory Multitarget Agents Acting as Dual Modulators of the Cannabinoid CB2 Receptor and Fatty Acid Amide Hydrolase. J Med Chem. 2023 Jan 12;66(1):235-250.?
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