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EX-A5386
CAS No. 2452396-89-1
EX-A5386( —— )
Catalog No. M35951 CAS No. 2452396-89-1
EX-A5386 (Glucocorticoid receptor modulator-1) is a potent glucocorticoid receptor modulator, IC50/EC50<100nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 202 | In Stock |
|
| 10MG | 306 | In Stock |
|
| 25MG | 511 | In Stock |
|
| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameEX-A5386
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NoteResearch use only, not for human use.
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Brief DescriptionEX-A5386 (Glucocorticoid receptor modulator-1) is a potent glucocorticoid receptor modulator, IC50/EC50<100nM.
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DescriptionGlucocorticoid receptor modulator 2 (Example 1) is a glucocorticoid receptor modulator, with an IC50 value less than 100 nM. Glucocorticoid receptor modulator 2 can be used for research of inflammatory and immune diseases.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayOthers
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TargetOther Targets
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RecptorGlucocorticoid Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number2452396-89-1
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Formula Weight482.55
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Molecular FormulaC29H27FN4O2
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Purity>98% (HPLC)
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Solubility——
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SMILESN(C(=O)C1CC1)[C@@H]2[C@H](N(C(=O)C2(C)C)C=3C=C4C(=CC3)N(N=C4)C5=CC=C(F)C=C5)C6=CC=CC=C6
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Florian JAKOB, et al. Substituted pyrrolidine amides iii. Patent. WO2020144375.
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