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Tyrphostin AG 538
CAS No. 133550-18-2
Tyrphostin AG 538( —— )
Catalog No. M35935 CAS No. 133550-18-2
Tyrphostin AG 538 is a chalcone compound, an IGF-1 receptor kinase inhibitor (IC 0 : for 400 nM) that is potent, cell-permeable, reversible, and competitive.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 152 | Get Quote |
|
| 5MG | 235 | Get Quote |
|
| 10MG | 353 | Get Quote |
|
| 25MG | 601 | Get Quote |
|
| 50MG | 821 | Get Quote |
|
| 100MG | 1062 | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameTyrphostin AG 538
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NoteResearch use only, not for human use.
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Brief DescriptionTyrphostin AG 538 is a chalcone compound, an IGF-1 receptor kinase inhibitor (IC 0 : for 400 nM) that is potent, cell-permeable, reversible, and competitive.
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DescriptionAG 538 is a potent, competitive inhibitor of IGF-1 receptor kinase, with an IC50 of 400 nM.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayAngiogenesis
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TargetIGF-1R
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RecptorIGF-1R
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Research Area——
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Indication——
Chemical Information
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CAS Number133550-18-2
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Formula Weight297.26
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Molecular FormulaC16H11NO5
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Purity>98% (HPLC)
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Solubility——
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SMILESC(/C(=C/C1=CC(O)=C(O)C=C1)/C#N)(=O)C2=CC(O)=C(O)C=C2
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. G Blum, et al. Substrate Competitive Inhibitors of IGF-1 Receptor Kinase. Biochemistry. 2000 Dec 26;39(51):15705-12.?
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