Tyrphostin AG 538

CAS No. 133550-18-2

Tyrphostin AG 538( —— )

Catalog No. M35935 CAS No. 133550-18-2

Tyrphostin AG 538 is a chalcone compound, an IGF-1 receptor kinase inhibitor (IC 0 : for 400 nM) that is potent, cell-permeable, reversible, and competitive.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 193 In Stock
10MG 292 In Stock
25MG 513 In Stock
50MG 686 In Stock
100MG 909 In Stock
200MG Get Quote In Stock
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Biological Information

  • Product Name
    Tyrphostin AG 538
  • Note
    Research use only, not for human use.
  • Brief Description
    Tyrphostin AG 538 is a chalcone compound, an IGF-1 receptor kinase inhibitor (IC 0 : for 400 nM) that is potent, cell-permeable, reversible, and competitive.
  • Description
    AG 538 is a potent, competitive inhibitor of IGF-1 receptor kinase, with an IC50 of 400 nM.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Angiogenesis
  • Target
    IGF-1R
  • Recptor
    IGF-1R
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    133550-18-2
  • Formula Weight
    297.26
  • Molecular Formula
    C16H11NO5
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    C(/C(=C/C1=CC(O)=C(O)C=C1)/C#N)(=O)C2=CC(O)=C(O)C=C2
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. G Blum, et al. Substrate Competitive Inhibitors of IGF-1 Receptor Kinase. Biochemistry. 2000 Dec 26;39(51):15705-12.?
molnova catalog
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