USP1-IN-2

CAS No. 2098212-05-4

USP1-IN-2( —— )

Catalog No. M35724 CAS No. 2098212-05-4

USP1-IN-2 is a potent USP1 inhibitor with potential anti-tumor activity for the study of cancer.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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5MG 686 In Stock
10MG 905 In Stock
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Biological Information

  • Product Name
    USP1-IN-2
  • Note
    Research use only, not for human use.
  • Brief Description
    USP1-IN-2 is a potent USP1 inhibitor with potential anti-tumor activity for the study of cancer.
  • Description
    USP1-IN-2 (Compound I-193) is a potent ubiquitin-specific protease 1 (USP1) inhibitor with an IC50 of less than about 50 nM.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Proteasome/Ubiquitin
  • Target
    DUB
  • Recptor
    DUB
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2098212-05-4
  • Formula Weight
    510.486
  • Molecular Formula
    C26H22F4N6O
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 62.5 mg/mL (122.43 mM; Ultrasonic (<60°C)
  • SMILES
    CC(C)c1c(F)cccc1-c1ncc2[nH]c(=O)n(Cc3ccc(cc3)-c3nc(cn3C)C(F)(F)F)c2n1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Alexandre Joseph Buckmelter, et al. Purinones as ubiquitin-specific protease 1 inhibitors. Patent US20170145012A1.
molnova catalog
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