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USP1-IN-2
CAS No. 2098212-05-4
USP1-IN-2( —— )
Catalog No. M35724 CAS No. 2098212-05-4
USP1-IN-2 is a potent USP1 inhibitor with potential anti-tumor activity for the study of cancer.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 445 | Get Quote |
|
| 5MG | 686 | Get Quote |
|
| 10MG | 905 | Get Quote |
|
| 25MG | 1334 | Get Quote |
|
| 50MG | 1730 | Get Quote |
|
| 100MG | 2313 | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameUSP1-IN-2
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NoteResearch use only, not for human use.
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Brief DescriptionUSP1-IN-2 is a potent USP1 inhibitor with potential anti-tumor activity for the study of cancer.
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DescriptionUSP1-IN-2 (Compound I-193) is a potent ubiquitin-specific protease 1 (USP1) inhibitor with an IC50 of less than about 50 nM.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayProteasome/Ubiquitin
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TargetDUB
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RecptorDUB
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Research Area——
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Indication——
Chemical Information
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CAS Number2098212-05-4
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Formula Weight510.486
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Molecular FormulaC26H22F4N6O
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 62.5 mg/mL (122.43 mM; Ultrasonic (<60°C)
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SMILESCC(C)c1c(F)cccc1-c1ncc2[nH]c(=O)n(Cc3ccc(cc3)-c3nc(cn3C)C(F)(F)F)c2n1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Alexandre Joseph Buckmelter, et al. Purinones as ubiquitin-specific protease 1 inhibitors. Patent US20170145012A1.
molnova catalog
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