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hGPR91 antagonist 3

CAS No. 1314796-31-0

hGPR91 antagonist 3( —— )

Catalog No. M35675 CAS No. 1314796-31-0

hGPR91 antagonist 3 is an orally active, potent, and selective hGPR91 antagonist. hGPR91 antagonist 3 is used to study hypertension, autoimmune diseases, and retinal angiogenesis.

Purity : >98% (HPLC)

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Datasheet

HNMR

HPLC

MSDS

Handing Instructions

Size	Price / USD	Stock	Quantity
1 mL x 10 mM in DMSO	315	In Stock
5MG	312	In Stock
10MG	518	In Stock
25MG	835	In Stock
50MG	1107	In Stock
100MG	1516	In Stock
200MG	2037	In Stock
500MG	Get Quote	In Stock
1G	Get Quote	In Stock

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Biological Information

Product Name

hGPR91 antagonist 3
Note

Research use only, not for human use.
Brief Description

hGPR91 antagonist 3 is an orally active, potent, and selective hGPR91 antagonist. hGPR91 antagonist 3 is used to study hypertension, autoimmune diseases, and retinal angiogenesis.
Description

hGPR91 antagonist 3 (Compound 5g) is a potent and orally active GPR91 antagonist with IC50 of 35 nM and 135 nM, for human GPR91 and rat GPR91, respectively.
In Vitro

——
In Vivo

——
Synonyms

——
Pathway

Cell Cycle/DNA Damage
Target

GPR
Recptor

GPR
Research Area

——
Indication

——

Chemical Information

CAS Number

1314796-31-0
Formula Weight

458.41
Molecular Formula

C23H18F4N4O2
Purity

>98% (HPLC)
Solubility

In Vitro:?DMSO : 100 mg/mL (218.15 mM; Ultrasonic (<80°C)
SMILES

O=C(NCC=1ON=C(C1)C=2C=CC(F)=C(C2)C(F)(F)F)CCCC=3N=C4N=CC=CC4=CC3
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. Bhuniya D, et al. Discovery of a potent and selective small molecule hGPR91 antagonist. Bioorg Med Chem Lett. 2011;21(12):3596-3602. ?

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