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GLP-1R modulator C5
CAS No. 421578-93-0
GLP-1R modulator C5( —— )
Catalog No. M35562 CAS No. 421578-93-0
GLP-1R modulator C5 is a small molecule GLP-1R orthosteric modulator that enhances GLP-1 binding to GLP-1R via transmembrane sites and can be used in the study of type II diabetes.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 53 | In Stock |
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| 100MG | Get Quote | In Stock |
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| 200MG | Get Quote | In Stock |
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| 500MG | Get Quote | In Stock |
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Biological Information
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Product NameGLP-1R modulator C5
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NoteResearch use only, not for human use.
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Brief DescriptionGLP-1R modulator C5 is a small molecule GLP-1R orthosteric modulator that enhances GLP-1 binding to GLP-1R via transmembrane sites and can be used in the study of type II diabetes.
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DescriptionGLP-1R modulator C5 is an allosteric modulator enhancing GLP-1 binding to GLP-1R via a transmembrane site (EC50 1.59 ± 0.53 μM).
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayGPCR/G Protein
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TargetGlucagon Receptor
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RecptorGlucagon Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number421578-93-0
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Formula Weight371.43
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Molecular FormulaC24H21NO3
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 50 mg/mL (134.61 mM; Ultrasonic )
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SMILESOC1(CC(=O)c2ccccc2)C(=O)N(CCc2ccccc2)c2ccccc12
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Wang J, et al. Allosteric Modulators Enhancing GLP-1 Binding to GLP-1R via a Transmembrane Site. ACS Chem Biol. 2021 Nov 19;16(11):2444-2452. ?
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