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FGFR2-IN-1

CAS No. 2677709-76-9

FGFR2-IN-1( —— )

Catalog No. M35540 CAS No. 2677709-76-9

FGFR2-IN-1 is an FGFR inhibitor that inhibits FGFR1, FGFR2, and FGFR3 with IC50s of 460, 140, and 2200 nM, respectively.FGFR2-IN-1 can be used for the study of cancers associated with FGFR2.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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25MG 158 In Stock
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Biological Information

  • Product Name
    FGFR2-IN-1
  • Note
    Research use only, not for human use.
  • Brief Description
    FGFR2-IN-1 is an FGFR inhibitor that inhibits FGFR1, FGFR2, and FGFR3 with IC50s of 460, 140, and 2200 nM, respectively.FGFR2-IN-1 can be used for the study of cancers associated with FGFR2.
  • Description
    FGFR2-IN-1 is a selective FGFR2 inhibitor with an IC50 of 140 nM.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Angiogenesis
  • Target
    FGFR
  • Recptor
    FGFR
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2677709-76-9
  • Formula Weight
    357.41
  • Molecular Formula
    C22H19N3O2
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    O=C(NC1=NNC=2C=C(C=CC12)C=3C=CC=C(OCC)C3)C=4C=CC=CC4
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Turner LD, et al. From Fragment to Lead: De Novo Design and Development toward a Selective FGFR2 Inhibitor. J. Med. Chem. 2021 Nov 15.
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