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PKA-IN-1
CAS No. 179985-52-5
PKA-IN-1( —— )
Catalog No. M35100 CAS No. 179985-52-5
PKA-IN-1 is a selective and potent cyclic AMP-dependent protein kinase (PKA) catalytic subunit (cAK) inhibitor (IC50: 0.03 μM).PKA-IN-1 can be used to study diseases of the immune system.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 66 | In Stock |
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| 10MG | 37 | In Stock |
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| 25MG | 61 | In Stock |
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| 50MG | 91 | In Stock |
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| 100MG | 144 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
|
Biological Information
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Product NamePKA-IN-1
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NoteResearch use only, not for human use.
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Brief DescriptionPKA-IN-1 is a selective and potent cyclic AMP-dependent protein kinase (PKA) catalytic subunit (cAK) inhibitor (IC50: 0.03 μM).PKA-IN-1 can be used to study diseases of the immune system.
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DescriptionPKA-IN-1 is a potent and selective cyclic AMP-dependent protein kinase (PKA) catalytic subunit (cAK) inhibitor with an IC50 of 0.03 μM.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayApoptosis
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TargetPKA
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RecptorPKA
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Research Area——
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Indication——
Chemical Information
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CAS Number179985-52-5
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Formula Weight225.25
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Molecular FormulaC13H11N3O
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 62.5 mg/mL (277.47 mM; Ultrasonic (<80°C)
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SMILESCC(=O)Nc1nc(C)c(C#N)c2ccccc12
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Z X Lu, et al. Selective inhibition of cyclic AMP-dependent protein kinase by isoquinoline derivative. Biol Chem Hoppe Seyler. 1996 Jun;377(6):373-8?
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