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Xanomeline tartrate
CAS No. 152854-19-8
Xanomeline tartrate( —— )
Catalog No. M35083 CAS No. 152854-19-8
Xanomeline tartrate (LY 246708 tartrate) is an M1 and M4 mAChR agonist with antipsychotic-like activity that improves cognition and can be used in studies of schizophrenia and Alzheimer's disease.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 29 | In Stock |
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| 5MG | 44 | In Stock |
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| 10MG | 61 | In Stock |
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| 25MG | 93 | In Stock |
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| 50MG | 138 | In Stock |
|
| 100MG | 202 | In Stock |
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| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameXanomeline tartrate
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NoteResearch use only, not for human use.
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Brief DescriptionXanomeline tartrate (LY 246708 tartrate) is an M1 and M4 mAChR agonist with antipsychotic-like activity that improves cognition and can be used in studies of schizophrenia and Alzheimer's disease.
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DescriptionXanomeline (LY 246708) is the potent agonist of muscarinic M1/M4 receptor with antipsychotic-like activity. Xanomeline (LY 246708) increases neuronal excitability.Xanomeline (LY 246708) can be used for the research of schizophrenia.
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In Vitro——
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In VivoAnimal Model:Male Cebus apella monkeys Dosage:0.5-3 mg/kg Administration:s.c.; 1-3 hours Result:Induced salivation and vomiting in some monkeys.
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Synonyms——
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PathwayOthers
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TargetOther Targets
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RecptorOthers
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Research Area——
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Indication——
Chemical Information
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CAS Number152854-19-8
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Formula Weight431.5
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Molecular FormulaC18H29N3O7S
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 250 mg/mL (579.37 mM; Ultrasonic )
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SMILESO[C@@H]([C@H](O)C(O)=O)C(O)=O.CCCCCCOc1nsnc1C1=CCCN(C)C1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Kreir M, et al. Role of Kv7.2/Kv7.3 and M1 muscarinic receptors in the regulation of neuronal excitability in hiPSC-derived neurons. Eur J Pharmacol. 2019;858:172474. ?
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