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Vazegepant
CAS No. 1337918-83-8
Vazegepant( —— )
Catalog No. M35066 CAS No. 1337918-83-8
Vazegepant (Zavegepant) is an orally available and selective antagonist of the calcitonin gene-related peptide CGRP receptor for pain relief and may be used in the study of migraine.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 306 | Get Quote |
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| 5MG | 227 | Get Quote |
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| 10MG | 335 | Get Quote |
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| 25MG | 567 | Get Quote |
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| 50MG | 792 | Get Quote |
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| 100MG | 1088 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameVazegepant
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NoteResearch use only, not for human use.
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Brief DescriptionVazegepant (Zavegepant) is an orally available and selective antagonist of the calcitonin gene-related peptide CGRP receptor for pain relief and may be used in the study of migraine.
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DescriptionVazegepant (Zavegepant) is an orally active calcitonin gene-related peptideCGRP receptor antagonist with potential for acute research in migraine. CGRP is an important trigger in migraine pathophysiology.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayGPCR/G Protein
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TargetCGRP Receptor
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RecptorCGRP Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number1337918-83-8
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Formula Weight638.8
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Molecular FormulaC36H46N8O3
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Purity>98% (HPLC)
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Solubility——
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SMILESO=C1C(=CC=2C(N1)=CC=CC2)C3CCN(C(N[C@H](CC=4C=C5C(=C(C)C4)NN=C5)C(=O)N6CCN(CC6)C7CCN(C)CC7)=O)CC3
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Leonard KA, et al. Discovery of a Gut-Restricted JAK Inhibitor for the Treatment of Inflammatory Bowel Disease. J Med Chem. 2020 Mar 26;63(6):2915-2929.?
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