Atogepant

CAS No. 1374248-81-3

Atogepant( MK-8031 | AGN-241689 )

Catalog No. M11545 CAS No. 1374248-81-3

A potent, selective and orally available CGRP receptor antagonist for the prevention of migraine.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 353 In Stock
5MG 264 In Stock
10MG 330 In Stock
25MG 655 In Stock
50MG 1144 In Stock
100MG 1665 In Stock
200MG 2251 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Atogepant
  • Note
    Research use only, not for human use.
  • Brief Description
    A potent, selective and orally available CGRP receptor antagonist for the prevention of migraine.
  • Description
    A potent, selective and orally available CGRP receptor antagonist for the prevention of migraine.Migraine Phase 3 Clinical.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    MK-8031 | AGN-241689
  • Pathway
    GPCR/G Protein
  • Target
    CGRP Receptor
  • Recptor
    CGRP Receptor
  • Research Area
    Neurological Disease
  • Indication
    Migraine

Chemical Information

  • CAS Number
    1374248-81-3
  • Formula Weight
    603.525
  • Molecular Formula
    C29H23F6N5O3
  • Purity
    >98% (HPLC)
  • Solubility
    10 mM in DMSO
  • SMILES
    O=C(C1=CN=C2C(C[C@@]3(C4=CC=CN=C4NC3=O)C2)=C1)N[C@@H]5C(N(CC(F)(F)F)[C@H](C)[C@H](C6=C(F)C=CC(F)=C6F)C5)=O
  • Chemical Name
    (3'S)-N-[(3S,5S,6R)-6-methyl-2-oxo-1-(2,2,2-trifluoroethyl)-5-(2,3,6-trifluorophenyl)piperidin-3-yl]-2'-oxo-1',2',5,7-tetrahydrospiro[cyclopenta[b]pyridine-6,3'-pyrrolo[2,3-b]pyridine]-3-carboxamide

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

molnova catalog
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