Cart
sales@molnova.com
EZM0414 TFA
CAS No. 2411759-92-5
EZM0414 TFA( —— )
Catalog No. M34899 CAS No. 2411759-92-5
EZM0414 TFA (SETD2-IN-1 TFA) is a SETD2 inhibitor with anticancer and antiproliferative effects for the study of leukemia and immune dysfunction.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 243 | Get Quote |
|
| 100MG | Get Quote | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
-
Product NameEZM0414 TFA
-
NoteResearch use only, not for human use.
-
Brief DescriptionEZM0414 TFA (SETD2-IN-1 TFA) is a SETD2 inhibitor with anticancer and antiproliferative effects for the study of leukemia and immune dysfunction.
-
DescriptionEZM0414 TFA is a potent, selective and orally active inhibitor of SETD2 which is a human histone methyltransferase. EZM0414 TFA has anti-proliferative effects.
-
In Vitro——
-
In Vivo——
-
Synonyms——
-
PathwayOthers
-
TargetOther Targets
-
RecptorHistone Methyltransferase
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number2411759-92-5
-
Formula Weight514.51
-
Molecular FormulaC24H30F4N4O4
-
Purity>98% (HPLC)
-
SolubilityIn Vitro:?DMSO : 200 mg/mL (388.72 mM; Ultrasonic ) H2O : 6.67 mg/mL (12.96 mM; Ultrasonic (<60°C))
-
SMILESOC(=O)C(F)(F)F.CC(=O)N1CCN(CC1)[C@H]1CCC[C@H](C1)NC(=O)c1cc2c(F)ccc(C)c2[nH]1
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. John Lampe, et al. Substituted indoles and methods of use thereof. WO2020037079A1.
molnova catalog
related products
-
Acacetin7-O-glucuron...
Acacetin 7-O-glucuronide is a glucuronide isolated from the methanolic leaf extract of Acacetin. Acacetin 7-O-glucuronide has potential applications in the development of nutraceuticals and pharmaceutical formulations.
-
Sivifene
Sivifene can be used for research on the treatment of cutaneous metastases from cancer.
-
1,3,6-Trihydroxy-2-m...
1,3,6-Trihydroxy-2-methylanthraquinone 3-O-(6'-O-acetyl)-alpha-L-rhamnosyl-(1->2)-Beta-D-glucoside shows certain antibacterial activity.
