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JAK1-IN-8
CAS No. 1973485-18-5
JAK1-IN-8( —— )
Catalog No. M34801 CAS No. 1973485-18-5
JAK1-IN-8, a specific inhibitor of Janus kinase 1 (JAK1, IC50<500 nM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 41 | In Stock |
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| 5MG | 37 | In Stock |
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| 10MG | 68 | In Stock |
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| 25MG | 140 | In Stock |
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| 50MG | 245 | In Stock |
|
| 100MG | 416 | In Stock |
|
| 200MG | 556 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameJAK1-IN-8
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NoteResearch use only, not for human use.
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Brief DescriptionJAK1-IN-8, a specific inhibitor of Janus kinase 1 (JAK1, IC50<500 nM).
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DescriptionJAK1-IN-8, a potent JAK1 inhibitor (IC50<500 nM), compound 28, extracted from patent WO2016119700A1.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayAngiogenesis
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TargetJAK
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RecptorJAK
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Research Area——
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Indication——
Chemical Information
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CAS Number1973485-18-5
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Formula Weight442.51
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Molecular FormulaC22H23FN4O3S
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 125 mg/mL (282.48 mM; Ultrasonic )
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SMILESFc1cc(ccc1CN1CCS(=O)(=O)CC1)-c1cccc2nc(NC(=O)C3CC3)cn12
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Jin Li, et al. Composés d'imidazo[1,2-a]pyridin-2-ylamine substitués, compositions pharmaceutiques et leurs méthodes d'utilisation. Patent WO2016119700A1.
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