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Home - Products - GPCR/G Protein - Cannabinoid Receptor - AZD1940

AZD1940

CAS No. 881413-29-2

AZD1940( —— )

Catalog No. M34518 CAS No. 881413-29-2

AZD1940 (UNII-0J0035E9FT) is a high affinity CB(1)/CB(2) receptor agonist of the cannabinoid with oral activity. Application in the study of orofacial pain.

Purity : >98% (HPLC)

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Biological Information

  • Product Name
    AZD1940
  • Note
    Research use only, not for human use.
  • Brief Description
    AZD1940 (UNII-0J0035E9FT) is a high affinity CB(1)/CB(2) receptor agonist of the cannabinoid with oral activity. Application in the study of orofacial pain.
  • Description
    AZD1940 is an orally active, high affinity cannabinoid CB1/CB2 receptor agonist with pKi values of 7.93 and 9.06 for human CB1R and CB2R, respectively. AZD1940 shows a robust analgesia action.
  • In Vitro
    AZD1940 binds with high affinity to human, rat and mouse CB1 and CB2 receptors and displays full agonism at both receptors in all three species.
  • In Vivo
    When given orally to rats, AZD1940 produces a robust analgesia in different models of inflammatory and neuropathic pain.For AZD1940, low brain uptake at analgesic doses has been demonstrated in both rats and primates.
  • Synonyms
    ——
  • Pathway
    GPCR/G Protein
  • Target
    Cannabinoid Receptor
  • Recptor
    Cannabinoid Receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    881413-29-2
  • Formula Weight
    413.52
  • Molecular Formula
    C20H29F2N3O2S
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 100 mg/mL (241.83 mM; Ultrasonic )
  • SMILES
    CCS(=O)(=O)Nc1ccc2n(CC3CCC(F)(F)CC3)c(nc2c1)C(C)(C)C
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Jarkko Kalliom?ki, et al. Evaluation of the analgesic efficacy and psychoactive effects of AZD1940, a novel peripherally acting cannabinoid agonist, in human capsaicin-induced pain and hyperalgesia. Clin Exp Pharmacol Physiol. 2013 Mar;40(3):212-8.?
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