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VRT-532
CAS No. 38214-71-0
VRT-532( —— )
Catalog No. M34468 CAS No. 38214-71-0
VRT-532 (CFpot-532) is an effective modulator of CFTR and is commonly used in studies of cystic fibrosis (CF) caused by CFTR defects.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 141 | In Stock |
|
| 5MG | 159 | In Stock |
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| 10MG | 238 | In Stock |
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| 25MG | 392 | In Stock |
|
| 50MG | 520 | In Stock |
|
| 100MG | 684 | In Stock |
|
| 200MG | 905 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameVRT-532
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NoteResearch use only, not for human use.
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Brief DescriptionVRT-532 (CFpot-532) is an effective modulator of CFTR and is commonly used in studies of cystic fibrosis (CF) caused by CFTR defects.
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DescriptionVRT-532 (CFpot-532) is a potent is a potent CFTR modulator. VRT-532 enhances channel activity in G551D-CFTR and intrinsic ATPase activity of G551D-CFTR. VRT-532 has the potential for the research of cystic fibrosis.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayApoptosis
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TargetCFTR
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RecptorCFTR
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Research Area——
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Indication——
Chemical Information
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CAS Number38214-71-0
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Formula Weight250.3
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Molecular FormulaC16H14N2O
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Purity>98% (HPLC)
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Solubility——
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SMILESCC1=CC=C(O)C(=C1)C1=NNC(=C1)C1=CC=CC=C1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Pasyk S, et al. Direct interaction of a small-molecule modulator with G551D-CFTR, a cystic fibrosis-causing mutation associated with severe disease. Biochem J. 2009 Feb 15;418(1):185-90. ?
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