Cart
sales@molnova.com
Tiospirone
CAS No. 87691-91-6
Tiospirone( —— )
Catalog No. M34041 CAS No. 87691-91-6
Tiospirone (BMY 13859-1 free base) is a 5-HT2 receptor antagonist and dopamine blocker that inhibits D2, 5-HT1a, 5-HT7, and sigma receptors.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 373 | In Stock |
|
| 5MG | 309 | In Stock |
|
| 10MG | 567 | In Stock |
|
| 25MG | 910 | In Stock |
|
| 50MG | 1200 | In Stock |
|
| 100MG | 1609 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
-
Product NameTiospirone
-
NoteResearch use only, not for human use.
-
Brief DescriptionTiospirone (BMY 13859-1 free base) is a 5-HT2 receptor antagonist and dopamine blocker that inhibits D2, 5-HT1a, 5-HT7, and sigma receptors.
-
DescriptionTiospirone is a 5-HT2 receptor antagonist with affinity for D2, 5-HT1a, and 5-HT7, and sigma receptors. Tiospirone decreases consumption of ethanol while increasing food intake of rats. Tiospirone can also reduce the reinforcing properties of Cocaine exhibited in the conditioned place preference paradigm.
-
In Vitro——
-
In Vivo——
-
Synonyms——
-
PathwayGPCR/G Protein
-
TargetDopamine Receptor
-
RecptorDopamine Receptor | 5-HT Receptor
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number87691-91-6
-
Formula Weight440.6
-
Molecular FormulaC24H32N4O2S
-
Purity>98% (HPLC)
-
Solubility——
-
SMILESO=C1N(C(=O)CC2(C1)CCCC2)CCCCN3CCN(C4=NSC=5C=CC=CC54)CC3
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Arolfo MP, et, al. Effects of amperozide and tiospirone, atypical antipsychotic 5-HT2 drugs, on food-reinforced behavior in rats. Physiol Behav. 1999 Dec;68(1-2):93-8.?
molnova catalog
related products
-
Trimethobenzamide hy...
Trimethobenzamide hydrochloride is a blocker of the D2 receptor. Trimethobenzamide is an antiemetic used to prevent nausea and vomiting.
-
Domperidone
Domperidone(Motilium) is a dopamine blocker and an antidopaminergic reagent.
-
FIIN-2
FIIN-2, an irreversible, pan-FGFR inhibitor, inhibits FGFR1/2/3/4 with IC50 of 3.09 nM, 4.3 nM, 27 nM and 45.3 nM, respectively.
