SCH 221510

CAS No. 322473-89-2

SCH 221510( —— )

Catalog No. M33925 CAS No. 322473-89-2

SCH 221510 is an orally available, selective and potent NOP agonist with an EC50 of 12 nM and a Ki of 0.3 nM.SCH 221510 has anxiolytic activity and can be used to study neurological disorders.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 163 In Stock
10MG 264 In Stock
25MG 534 In Stock
50MG 830 In Stock
100MG 1349 In Stock
200MG 1814 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    SCH 221510
  • Note
    Research use only, not for human use.
  • Brief Description
    SCH 221510 is an orally available, selective and potent NOP agonist with an EC50 of 12 nM and a Ki of 0.3 nM.SCH 221510 has anxiolytic activity and can be used to study neurological disorders.
  • Description
    SCH 221510 is a potent, orally active and selective NOP (nociceptin opioid receptor) agonist, with an EC50 of 12 nM and Ki of 0.3 nM. SCH 221510 shows an anxiolytic-like effect.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Endocrinology/Hormones
  • Target
    Opioid Receptor
  • Recptor
    Opioid Receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    322473-89-2
  • Formula Weight
    397.55
  • Molecular Formula
    C28H31NO
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    C(N1[C@@]2(C[C@@](O)(C[C@]1(CC2)[H])C3=CC=CC=C3)[H])(C4=C(C)C=CC=C4)C5=C(C)C=CC=C5
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Varty GB, et al. The anxiolytic-like effects of the novel, orally active nociceptin opioid receptor agonist 8-[bis(2-methylphenyl)methyl]-3-phenyl-8-azabicyclo[3.2.1]octan-3-ol (SCH 221510). J Pharmacol Exp Ther. 2008 Aug;326(2):672-82.?
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