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BMS 753
CAS No. 215307-86-1
BMS 753( —— )
Catalog No. M33783 CAS No. 215307-86-1
BMS 753 is an agonist of isotype-selective retinoic acid receptor α (RARα, Ki= 2 nM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 55 | In Stock |
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| 5MG | 55 | In Stock |
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| 10MG | 92 | In Stock |
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| 25MG | 212 | In Stock |
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| 50MG | 333 | In Stock |
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| 100MG | 462 | In Stock |
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| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameBMS 753
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NoteResearch use only, not for human use.
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Brief DescriptionBMS 753 is an agonist of isotype-selective retinoic acid receptor α (RARα, Ki= 2 nM).
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DescriptionBMS 753 is an isotype-selective retinoic acid receptor α (RARα) agonist, with a Ki of 2 nM.
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In VitroBMS 753 results in low levels of RARβ transcripts in WT cells, RARγ-/-, but not activates in RARa-/- cells.
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In Vivo——
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Synonyms——
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PathwayMetabolic Enzyme/Protease
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TargetRetinoid Receptor
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RecptorRetinoid Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number215307-86-1
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Formula Weight351.4
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Molecular FormulaC21H21NO4
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 50 mg/mL (142.29 mM; Ultrasonic )
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SMILESCC1(C)C(=O)C(C)(C)c2cc(ccc12)C(=O)Nc1ccc(cc1)C(O)=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. M Géhin, et al. Structural basis for engineering of retinoic acid receptor isotype-selective agonists and antagonists. Chem Biol. 1999 Aug;6(8):519-29.?
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