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Tyrphostin A25
CAS No. 118409-58-8
Tyrphostin A25( —— )
Catalog No. M33749 CAS No. 118409-58-8
Tyrphostin A25 (Tyrphostin AG 82) is a specific EGFR tyrosine kinase inhibitor and GPR35 agonist with an IC50 value of 0.94 μM for GPR35 and an EC50 value of 5.3 μM for GPR35.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 31 | In Stock |
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| 5MG | 49 | In Stock |
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| 10MG | 71 | In Stock |
|
| 25MG | 117 | In Stock |
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| 50MG | 169 | In Stock |
|
| 100MG | 250 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameTyrphostin A25
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NoteResearch use only, not for human use.
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Brief DescriptionTyrphostin A25 (Tyrphostin AG 82) is a specific EGFR tyrosine kinase inhibitor and GPR35 agonist with an IC50 value of 0.94 μM for GPR35 and an EC50 value of 5.3 μM for GPR35.
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DescriptionTyrphostin 25 (AG82) is a specific inhibitor of the EGFR tyrosine kinase. Tyrphostin 25 is also a GPR35 agonist with an IC50 of 0.94 μM and an EC50 of 5.3 μM.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayAngiogenesis
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TargetEGFR
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RecptorEGFR | GPR
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Research Area——
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Indication——
Chemical Information
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CAS Number118409-58-8
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Formula Weight202.17
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Molecular FormulaC10H6N2O3
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Purity>98% (HPLC)
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Solubility——
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SMILESC(=C(C#N)C#N)C1=CC(O)=C(O)C(O)=C1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Klemke RL, et al. Receptor tyrosine kinase signaling required for integrin alpha v beta 5-directed cell motility but not adhesion on vitronectin. J Cell Biol. 1994 Nov;127(3):859-66. ?
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