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CCT129957
CAS No. 883098-58-6
CCT129957( —— )
Catalog No. M33309 CAS No. 883098-58-6
CCT129957 is a novel and potent phospholipase C-γ (PLC-γ) inhibitor with an IC50 of about 3 μM and a GC50 of 15 μM.CCT129957 exhibits anticancer activity and inhibits Ca2+ release in squamous cells.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 93 | In Stock |
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| 5MG | 85 | In Stock |
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| 10MG | 128 | In Stock |
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| 25MG | 233 | In Stock |
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| 50MG | 341 | In Stock |
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| 100MG | 513 | In Stock |
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| 200MG | Get Quote | In Stock |
|
| 500MG | 1088 | In Stock |
|
| 1G | Get Quote | In Stock |
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Biological Information
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Product NameCCT129957
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NoteResearch use only, not for human use.
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Brief DescriptionCCT129957 is a novel and potent phospholipase C-γ (PLC-γ) inhibitor with an IC50 of about 3 μM and a GC50 of 15 μM.CCT129957 exhibits anticancer activity and inhibits Ca2+ release in squamous cells.
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DescriptionCCT129957 is an indole derivative and a potent phospholipase C-γ (PLC-γ) inhibitor with an IC50 of ~3 μM and a GC50 of 15 μM. CCT129957 inhibits Ca2+ release in squamous carcinoma cells at ~15 μM.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayMetabolic Enzyme/Protease
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TargetPhospholipase
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RecptorPhospholipase | Calcium Channel
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Research Area——
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Indication——
Chemical Information
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CAS Number883098-58-6
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Formula Weight309.32
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Molecular FormulaC17H15N3O3
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 100 mg/mL (323.29 mM; Ultrasonic )
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SMILES[O-][N+](=O)c1cccc2cc([nH]c12)C(=O)NCCc1ccccc1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
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PHPS1
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Abbolactone
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Melittin TFA(20449-7...
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