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ICI 174,864
CAS No. 89352-67-0
ICI 174,864( —— )
Catalog No. M30662 CAS No. 89352-67-0
Selective δ opioid antagonist. Exhibits partial agonist in vitro activity at δ receptors at high concentrations.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 10MG | 387 | Get Quote |
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| 100MG | Get Quote | Get Quote |
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| 200MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
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Biological Information
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Product NameICI 174,864
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NoteResearch use only, not for human use.
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Brief DescriptionSelective δ opioid antagonist. Exhibits partial agonist in vitro activity at δ receptors at high concentrations.
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DescriptionSelective δ opioid antagonist. Exhibits partial agonist in vitro activity at δ receptors at high concentrations.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayEndocrinology/Hormones
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TargetOpioid Receptor
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Recptor——
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Research Area——
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Indication——
Chemical Information
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CAS Number89352-67-0
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Formula Weight691.87
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Molecular FormulaC38H53N5O7
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Purity>98% (HPLC)
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SolubilityDMSO:69.19 mg/mL;water:1 mg/ml
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SMILESCC(C)C[C@H](NC(=O)[C@H](CC1=CC=CC=C1)NC(=O)C(C)(C)NC(=O)C(C)(C)NC(=O)[C@H](CC1=CC=C(O)C=C1)N(CC=C)CC=C)C(O)=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Cohen et al (1996) Opioid agonist activity of ICI 174864 and its carboxypeptidase degradation product, LY281217. J.Pharmacol.Exp.Ther. 238 769 PMID:
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