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c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2

CAS No. 1647119-61-6

c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2( —— )

Catalog No. M30172 CAS No. 1647119-61-6

c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 is a selective and short-acting peptidic V2 receptor (V2R) agonist with EC50s of 0.07nM and 0.02 nM for hV2R and rV2R, respectively.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2
  • Note
    Research use only, not for human use.
  • Brief Description
    c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 is a selective and short-acting peptidic V2 receptor (V2R) agonist with EC50s of 0.07nM and 0.02 nM for hV2R and rV2R, respectively.
  • Description
    c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 is a selective and short-acting peptidic V2 receptor (V2R) agonist with EC50s of 0.07nM and 0.02 nM for hV2R and rV2R, respectively.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    EC50: 0.07 nM (hV2R), 0.02 nM (rV2R)
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1647119-61-6
  • Formula Weight
    946.58
  • Molecular Formula
    C42H60ClN11O8S2
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    ——
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

Wi?niewski K, et al. Discovery of Potent, Selective, and Short-Acting Peptidic V2 Receptor Agonists. J Med Chem. 2019 May 23;62(10):4991-5005.
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