Atherosperminine

CAS No. 5531-98-6

Atherosperminine( Atherospermine )

Catalog No. M29285 CAS No. 5531-98-6

Atherosperminine shows cholinesterase inhibitory activity against acetylcholinesterase (AChE) and butyrylcholinesterase (BChE). Atherosperminine exerts a non-specific relaxant effect on the trachealis, its major mechanism of action appears to be inhibition of cAMP phosphodiesterase.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 211 In Stock
2MG 136 In Stock
5MG 208 In Stock
10MG 313 In Stock
25MG 534 In Stock
50MG 735 In Stock
100MG Get Quote In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Atherosperminine
  • Note
    Research use only, not for human use.
  • Brief Description
    Atherosperminine shows cholinesterase inhibitory activity against acetylcholinesterase (AChE) and butyrylcholinesterase (BChE). Atherosperminine exerts a non-specific relaxant effect on the trachealis, its major mechanism of action appears to be inhibition of cAMP phosphodiesterase.
  • Description
    Atherosperminine shows cholinesterase inhibitory activity against acetylcholinesterase (AChE) and butyrylcholinesterase (BChE). Atherosperminine exerts a non-specific relaxant effect on the trachealis, its major mechanism of action appears to be inhibition of cAMP phosphodiesterase.(In Vitro):Atherosperminine shows strong anti-plasmodial activity against Plasmodium falciparum, with the IC50 value of 5.80 μM. Atherosperminine also shows antioxidant activity in a DPPH assay with the IC50 value of 54.53 ug/mL.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    Atherospermine
  • Pathway
    GPCR/G Protein
  • Target
    cAMP
  • Recptor
    cAMP
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    5531-98-6
  • Formula Weight
    309.4
  • Molecular Formula
    C20H23NO2
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    COc1cc(CCN(C)C)c2ccc3ccccc3c2c1OC
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

molnova catalog
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