HIF1-IN-3?

CAS No. 333314-79-7

HIF1-IN-3?( Benzenepropanamide, N-[(8-hydroxy-7-quinolinyl)(4-methoxyphenyl)methyl]- )

Catalog No. M28955 CAS No. 333314-79-7

HIF1-IN-3 is an effective inhibitor of HIF-1 (EC50 = 0.9 μM) and can be used in anticancer studies.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 46 In Stock
5MG 36 In Stock
10MG 55 In Stock
25MG 112 In Stock
50MG 207 In Stock
100MG 286 In Stock
200MG 414 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    HIF1-IN-3?
  • Note
    Research use only, not for human use.
  • Brief Description
    HIF1-IN-3 is an effective inhibitor of HIF-1 (EC50 = 0.9 μM) and can be used in anticancer studies.
  • Description
    HIF1-IN-3 is an effective inhibitor of HIF-1 (EC50 = 0.9 μM) and can be used in anticancer studies.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    Benzenepropanamide, N-[(8-hydroxy-7-quinolinyl)(4-methoxyphenyl)methyl]-
  • Pathway
    Angiogenesis
  • Target
    HIF/HIF Prolyl-hydroxylase
  • Recptor
    SIRT2
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    333314-79-7
  • Formula Weight
    412.5
  • Molecular Formula
    C26H24N2O3
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 125 mg/mL (303.04 mM)
  • SMILES
    O=C(NC(C1=CC=C2C=CC=NC2=C1O)C3=CC=C(OC)C=C3)CCC4=CC=CC=C4
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Schiedel M, et al. Structure-Based Development of an Affinity Probe for Sirtuin 2. Angew Chem Int Ed Engl. 2016 Feb 5;55(6):2252-6.
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