M4 mAChR agonist-1?

CAS No. 785705-53-5

M4 mAChR agonist-1?( 4-Piperidinecarboxamide, 1-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)- )

Catalog No. M28954 CAS No. 785705-53-5

M4 mAChR agonist-1 is an effective agonist of M4 mAChR (EC50 >10 μM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 37 In Stock
5MG 61 In Stock
10MG 92 In Stock
25MG 169 In Stock
50MG 269 In Stock
100MG 398 In Stock
200MG Get Quote In Stock
500MG 901 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    M4 mAChR agonist-1?
  • Note
    Research use only, not for human use.
  • Brief Description
    M4 mAChR agonist-1 is an effective agonist of M4 mAChR (EC50 >10 μM).
  • Description
    M4 mAChR agonist-1 is an effective agonist of M4 mAChR (EC50 >10 μM).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    4-Piperidinecarboxamide, 1-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)-
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    AChR
  • Recptor
    Parasite
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    785705-53-5
  • Formula Weight
    290.389
  • Molecular Formula
    C14H18N4OS
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 20 mg/mL (68.88 mMul)
  • SMILES
    CC1=C(C)C2=C(N=CN=C2S1)N1CCC(CC1)C(N)=O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.G?tz MG, et al. Aza-peptidyl Michael acceptors. A new class of potent and selective inhibitors of asparaginyl endopeptidases (legumains) from evolutionarily diverse pathogens. J Med Chem. 2008 May 8;51(9):2816-32.
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