M4 mAChR agonist-1?
CAS No. 785705-53-5
M4 mAChR agonist-1?( 4-Piperidinecarboxamide, 1-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)- )
Catalog No. M28954 CAS No. 785705-53-5
M4 mAChR agonist-1 is an effective agonist of M4 mAChR (EC50 >10 μM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 35 | Get Quote |
|
| 5MG | 58 | Get Quote |
|
| 10MG | 87 | Get Quote |
|
| 25MG | 160 | Get Quote |
|
| 50MG | 260 | Get Quote |
|
| 100MG | 385 | Get Quote |
|
| 500MG | 872 | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
-
Product NameM4 mAChR agonist-1?
-
NoteResearch use only, not for human use.
-
Brief DescriptionM4 mAChR agonist-1 is an effective agonist of M4 mAChR (EC50 >10 μM).
-
DescriptionM4 mAChR agonist-1 is an effective agonist of M4 mAChR (EC50 >10 μM).
-
In Vitro——
-
In Vivo——
-
Synonyms4-Piperidinecarboxamide, 1-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)-
-
PathwayCell Cycle/DNA Damage
-
TargetAChR
-
RecptorParasite
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number785705-53-5
-
Formula Weight290.389
-
Molecular FormulaC14H18N4OS
-
Purity>98% (HPLC)
-
SolubilityIn Vitro:?DMSO : 20 mg/mL (68.88 mMul)
-
SMILESCC1=C(C)C2=C(N=CN=C2S1)N1CCC(CC1)C(N)=O
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1.G?tz MG, et al. Aza-peptidyl Michael acceptors. A new class of potent and selective inhibitors of asparaginyl endopeptidases (legumains) from evolutionarily diverse pathogens. J Med Chem. 2008 May 8;51(9):2816-32.
molnova catalog
related products
-
(±)-Acetylcarnitine ...
(±)-Acetylcarnitine chloride (Acetyl dl-carnitine chloride) is a weak cholinergic agonist with neuroprotective properties and can be used in studies of neuritis.
-
Tarafenacin D-tartra...
Tarafenacin D-tartrate (SVT-40776 D-tartrate) is a selective and potent muscarinic acetylcholine M3 receptor antagonist used in the study of overactive bladder and bronchial disorders.
-
Lobelanidine
Lobelanidine (8,10-Diphenyllobelidiol), which can be extracted from the above-ground parts of Lobelia chinensis Lour and Lobelia tupa, is an analogue of lobeline and shows a moderate affinity for nAChR.
Cart
sales@molnova.com