M4 mAChR agonist-1?

CAS No. 785705-53-5

M4 mAChR agonist-1?( 4-Piperidinecarboxamide, 1-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)- )

Catalog No. M28954 CAS No. 785705-53-5

M4 mAChR agonist-1 is an effective agonist of M4 mAChR (EC50 >10 μM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 35 Get Quote
5MG 58 Get Quote
10MG 87 Get Quote
25MG 160 Get Quote
50MG 260 Get Quote
100MG 385 Get Quote
500MG 872 Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    M4 mAChR agonist-1?
  • Note
    Research use only, not for human use.
  • Brief Description
    M4 mAChR agonist-1 is an effective agonist of M4 mAChR (EC50 >10 μM).
  • Description
    M4 mAChR agonist-1 is an effective agonist of M4 mAChR (EC50 >10 μM).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    4-Piperidinecarboxamide, 1-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)-
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    AChR
  • Recptor
    Parasite
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    785705-53-5
  • Formula Weight
    290.389
  • Molecular Formula
    C14H18N4OS
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 20 mg/mL (68.88 mMul)
  • SMILES
    CC1=C(C)C2=C(N=CN=C2S1)N1CCC(CC1)C(N)=O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.G?tz MG, et al. Aza-peptidyl Michael acceptors. A new class of potent and selective inhibitors of asparaginyl endopeptidases (legumains) from evolutionarily diverse pathogens. J Med Chem. 2008 May 8;51(9):2816-32.
molnova catalog
related products
  • (±)-Acetylcarnitine ...

    (±)-Acetylcarnitine chloride (Acetyl dl-carnitine chloride) is a weak cholinergic agonist with neuroprotective properties and can be used in studies of neuritis.

  • Tarafenacin D-tartra...

    Tarafenacin D-tartrate (SVT-40776 D-tartrate) is a selective and potent muscarinic acetylcholine M3 receptor antagonist used in the study of overactive bladder and bronchial disorders.

  • Lobelanidine

    Lobelanidine (8,10-Diphenyllobelidiol), which can be extracted from the above-ground parts of Lobelia chinensis Lour and Lobelia tupa, is an analogue of lobeline and shows a moderate affinity for nAChR.