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M4 mAChR agonist-1?
CAS No. 785705-53-5
M4 mAChR agonist-1?( 4-Piperidinecarboxamide, 1-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)- )
Catalog No. M28954 CAS No. 785705-53-5
M4 mAChR agonist-1 is an effective agonist of M4 mAChR (EC50 >10 μM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 37 | In Stock |
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| 5MG | 61 | In Stock |
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| 10MG | 92 | In Stock |
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| 25MG | 169 | In Stock |
|
| 50MG | 269 | In Stock |
|
| 100MG | 398 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | 901 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameM4 mAChR agonist-1?
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NoteResearch use only, not for human use.
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Brief DescriptionM4 mAChR agonist-1 is an effective agonist of M4 mAChR (EC50 >10 μM).
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DescriptionM4 mAChR agonist-1 is an effective agonist of M4 mAChR (EC50 >10 μM).
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In Vitro——
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In Vivo——
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Synonyms4-Piperidinecarboxamide, 1-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)-
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PathwayCell Cycle/DNA Damage
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TargetAChR
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RecptorParasite
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Research Area——
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Indication——
Chemical Information
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CAS Number785705-53-5
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Formula Weight290.389
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Molecular FormulaC14H18N4OS
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 20 mg/mL (68.88 mMul)
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SMILESCC1=C(C)C2=C(N=CN=C2S1)N1CCC(CC1)C(N)=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.G?tz MG, et al. Aza-peptidyl Michael acceptors. A new class of potent and selective inhibitors of asparaginyl endopeptidases (legumains) from evolutionarily diverse pathogens. J Med Chem. 2008 May 8;51(9):2816-32.
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