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NGD-8243
CAS No. 573678-04-3
NGD-8243( N-[4-(trifluoromethyl)phenyl]-7-[3-(trifluoromethyl)pyridin-2-yl]quinazolin-4-amine | NGD8243 | NGD 8243 )
Catalog No. M28921 CAS No. 573678-04-3
NGD-8243 is a TRPV1 inhibitor and can be used in studies for prevention and treatment of cardiac hypertrophy.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 472 | In Stock |
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| 5MG | 415 | In Stock |
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| 10MG | 614 | In Stock |
|
| 25MG | 938 | In Stock |
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| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameNGD-8243
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NoteResearch use only, not for human use.
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Brief DescriptionNGD-8243 is a TRPV1 inhibitor and can be used in studies for prevention and treatment of cardiac hypertrophy.
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DescriptionNGD-8243 is a TRPV1 inhibitor and can be used in studies for prevention and treatment of cardiac hypertrophy.
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In Vitro——
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In Vivo——
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SynonymsN-[4-(trifluoromethyl)phenyl]-7-[3-(trifluoromethyl)pyridin-2-yl]quinazolin-4-amine | NGD8243 | NGD 8243
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PathwayMembrane Transporter/Ion Channel
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TargetTRP/TRPV Channel
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Recptor——
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Research Area——
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Indication——
Chemical Information
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CAS Number573678-04-3
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Formula Weight434.345
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Molecular FormulaC21H12F6N4
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Purity>98% (HPLC)
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Solubility——
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SMILESFC(F)(F)c1ccc(Nc2ncnc3cc(ccc23)-c2ncccc2C(F)(F)F)cc1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Xue Z, Yan R, Yang B. Phenylethanoid glycosides and phenolic glycosides from stem bark of Magnolia officinalis. Phytochemistry. 2016 Jul;127:50-62.
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