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Dazcapistat
CAS No. 2221010-42-8
Dazcapistat( —— )
Catalog No. M28849 CAS No. 2221010-42-8
Dazcapistat is a potent calpain inhibitor, with IC50s of <3 μM for calpain 1, calpain 2 and calpain 9, respectively.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 223 | In Stock |
|
| 5MG | 202 | In Stock |
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| 10MG | 306 | In Stock |
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| 25MG | 550 | In Stock |
|
| 50MG | 756 | In Stock |
|
| 100MG | 1051 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameDazcapistat
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NoteResearch use only, not for human use.
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Brief DescriptionDazcapistat is a potent calpain inhibitor, with IC50s of <3 μM for calpain 1, calpain 2 and calpain 9, respectively.
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DescriptionDazcapistat is a potent calpain inhibitor, with IC50s of <3 μM for calpain 1, calpain 2 and calpain 9, respectively.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayProteasome/Ubiquitin
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TargetCysteine Protease
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Recptornecrosis(MLKL)
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Research Area——
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Indication——
Chemical Information
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CAS Number2221010-42-8
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Formula Weight395.39
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Molecular FormulaC21H18FN3O4
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 100 mg/mL (252.92 mM)
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SMILESO=C(C1=C(C2=CC=CC=C2F)N=C(C)O1)NC(C(C(N)=O)=O)CC3=CC=CC=C3
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Dodo K, et al. Indolylmaleimide Derivative IM-17 Shows Cardioprotective Effects in Ischemia-Reperfusion Injury. ACS Med Chem Lett. 2018 Jan 29;9(3):182-187.
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